Cat. No.: X24-05-ZQ128
PI3K inhibitor PI-103 hydrochloride, Purity ≥98%
Synonym: 371935-79-4; PI 103 hydrochloride; PI103 hydrochloride; PI3K inhibitor
- CAS Number: 371935-79-4
- Compound CID: 16739368
Product Size
10 mg; 50 mg; 100 mg
Properties
Description
PI-103 hydrochloride is a potent compound that inhibits PI3 kinase activity. It targets ATM, ATR, DNA-PK, hsVPS34, mTORC1, mTORC2, p110α, p110β, p110δ, p110γ, and PI3KC2α.
Molecular Formula
C19H17ClN4O3
Targets
ATM: 920 nM; ATR: 850 nM; DNA-PK: 2 nM; hsVPS34: 2.3 nM; mTORC1: 20 nM; mTORC2: 83 nM; p110α: 8 nM; p110β: 88 nM; p110δ: 48 nM; p110γ: 150 nM; PI3KC2α: 1 μM
Identity
Confirmed by NMR/HPLC/MS.
Applications
PI-103 hydrochloride is a dual PI3K/mTOR inhibitor used to research anticancer mechanisms.
Related Products
Quick Links