Epigenetic reader domain inhibitor MS402, Purity ≥98%

Synonym: 1672684-68-2; MS-402; MS 402; Epigenetic reader domain inhibitor

CAS Number: 1672684-68-2
Compound CID: 90718189

Product Size

5 mg; 10 mg; 50 mg

Price

Datasheet

MSDS

Properties

Description

MS402 disrupts the function of proteins that recognize and bind specific epigenetic marks, affecting the interpretation of epigenetic signals. It targets BRD2-BD1, BRD2-BD2, BRD3-BD1, BRD3-BD2, BRD4-BD1, and BRD4-BD2.

Molecular Weight

370.83

Molecular Formula

C₂₀H₁₉ClN₂O₃

Targets

BRD2-BD1: 83 nM (Ki); BRD2-BD2: 240 nM (Ki); BRD3-BD1: 110 nM (Ki); BRD3-BD2: 200 nM (Ki); BRD4-BD1: 77 nM (Ki); BRD4-BD2: 718 nM (Ki)

Form

Lyophilized powder

Purity

Identity

Confirmed by NMR/HPLC/MS.

Applications

MS402 serves as a research tool to explore the involvement of bromodomains in disease and gene expression patterns.