Cat. No.: X24-05-ZQ594
PRMT inhibitor EPZ020411 hydrochloride, Purity ≥98%
Synonym: 2070015-25-5; EPZ-020411; EPZ 020411; Protein arginine methyltransferase inhibitor
- CAS Number: 2070015-25-5
- Compound CID: 119081410
Product Size
5 mg; 10 mg; 50 mg; 100 mg
Properties
Description
EPZ020411 hydrochloride, soluble in DMSO, water and ethanol, inhibits enzymes that methylate arginine residues in proteins, impacting signaling pathways and gene regulation. It targets PRMT1, PRMT6, and PRMT8.
Molecular Formula
C25H39ClN4O3
Targets
PRMT1: 0.119 μM; PRMT6: 0.01 μM; PRMT8: 0.223 μM
Solubility
DMSO: 86 mg/mL (166.81 mM); Water: 70 mg/mL (135.78 mM); Ethanol: 86 mg/mL (166.81 mM)
Identity
Confirmed by NMR/HPLC/MS.
Applications
EPZ020411 hydrochloride can be used to inhibit G9a/GLP histone methyltransferase in epigenomics.
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