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PROTAC degrader inhibitor, ARV-771, Purity ≥98%
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Cat. No.: X24-09-YM730

PROTAC degrader inhibitor, ARV-771, Purity ≥98%

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Synonym: 1949837-12-0; ARV771; ARV 771; (2S,4R)-1-[(2S)-2-[[2-[3-[2-[[2-[(9S)-7-(4-Chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; PROTAC degrader inhibitor

  • CAS Number: 1949837-12-0
  • Compound CID: 126619980
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Product Size
1 mg; 5 mg; 10 mg; 50 mg
Price
Datasheet
Datasheet
MSDS
MSDS
Properties
Description
ARV-771, soluble in DMSO and ethanol and insoluble in water, is an effective PROTAC inhibitor, that has the ability to prevent the pathway of PROTAC degrader. The molecular weight of the compound is 986.64, and its molecular formula is C49H60ClN9O7S2. It targets the BRD2(1), BRD2(2), BRD3(1), BRD3(2), BRD4(1) and BRD4(2).
Molecular Weight
986.64
Molecular Formula
C49H60ClN9O7S2
Targets
BRD2 (1)
Form
Lyophilized powder
Purity
≥98%
Impurities
Free from inappropriate visible particulates, foreign matter, discoloration, or other defects.
Solubility
In vitro: DMSO: 97 mg/mL (98.31 mM); Water: insoluble; Ethanol: 97 mg/mL (98.31 mM)
Identity
Confirmed by NMR/HPLC/MS.
Applications
ARV-771 can be studied extensively for its potential therapeutic applications in the treatment of castration-resistant prostate cancer (CRPC) by eliminating the androgen receptor, which drives tumor growth in these patients.
Publications
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