Properties
Description
Seltorexant inhibits the signaling pathway between G-protein-coupled receptors (GPCRs) and G proteins. It targets human OX2R, and rat OX2R.
Molecular Formula
C21H22FN7O
Targets
Human OX2R: 8.0 (pKi); Rat OX2R: 8.1 (pKi)
Applications
Seltorexant can be studied for its effect on blocking the action of orexin, a neuropeptide involved in the regulation of wakefulness and sleep.