Cat. No.: X24-06-ZQ445
FAK inhibitor Defactinib, Purity ≥98%
Synonym: 1073154-85-4; FAK inhibitor; VS-6063; VS 6063; VS6063; PF-04554878; PF04554878; PF04554878
- MDL: MFCD25977806
- CAS Number: 1073154-85-4
- Compound CID: 25117126
Product Size
5 mg; 10 mg; 50 mg; 100 mg
Properties
Description
Defactinib, soluble in warmed DMSO and insoluble in water and ethanol, is a FAK inhibitor that is used to block angiogenesis in diseases such as cancer.
Molecular Formula
C20H21F3N8O3S
Solubility
Warmed DMSO: 5 mg/mL (9.79 mM); Water: Insoluble; Ethanol: Insoluble
Identity
Confirmed by NMR/HPLC/MS.
Applications
Defactinib is used to inhibit focal adhesion kinase, with implications for cancer metastasis and treatment strategies.
Related Products
Quick Links