Cat. No.: X24-05-ZQ237
RSK inhibitor BI-D1870, Purity ≥98%
Synonym: 501437-28-1; BI-D1870; 2-((3,5-Difluoro-4-hydroxyphenyl)amino)-8-isopentyl-5,7-dimethyl-7,8-dihydropteridin-6(5H)-one; BI-D 1870; 2-(3,5-Difluoro-4-hydroxyanilino)-5,7-dimethyl-8-(3-methylbutyl)-7H-pteridin-6-one; RSK inhibitor
- CAS Number: 501437-28-1
- Compound CID: 25023738
Product Size
5 mg; 10 mg; 25 mg; 50 mg
Properties
Description
BI-D1870, soluble in DMSO and insoluble in ethanol and water, attenuates the activity of kinases involved in cell growth, survival, and proliferation, which can be utilized to inhibit tumor progression. It targets RSK1, RSK2, RSK3, and RSK4.
Molecular Formula
C19H23F2N5O2
Targets
RSK1; RSK2; RSK3; RSK4
Solubility
DMSO: 71 mg/mL (181.39 mM); Water: Insoluble; Ethanol: Insoluble
Identity
Confirmed by NMR/HPLC/MS.
Applications
BI-D1870 can be employed to study its effects on RSK kinase activity and downstream signaling events in cancer.
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