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Cat. No.: X24-05-ZQ051

PI3K inhibitor SAR245409, Purity ≥98%

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Synonym: 934493-76-2; Voxtalisib; XL765; SAR 245409; SAR-245409; XL 765; XL-765; PI3K inhibitor

  • CAS Number: 934493-76-2
  • Compound CID: 16123056
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Product Size
5 mg; 10 mg; 50 mg
Price
Datasheet
Datasheet
MSDS
MSDS
Properties
Description
SAR245409, soluble in DMSO and insoluble in ethanol and water, is a potent compound that inhibits PI3 kinase activity. It targets PI3Kα, PI3Kδ, DNA-PK, mTOR, PI3Kβ, and PI3Kγ.
Molecular Weight
270.29
Molecular Formula
C13H14N6O
Targets
PI3Kα: 39 nM; PI3Kδ: 43 nM; DNA-PK: 150 nM; mTOR: 157 nM; PI3Kβ: 113 nM; PI3Kγ: 9 nM
Form
Lyophilized powder
Purity
≥98%
Solubility
DMSO: 53 mg/mL (196.08 mM); Water: Insoluble; Ethanol: Insoluble
Identity
Confirmed by NMR/HPLC/MS.
Applications
SAR245409 can be used to explore dual inhibition of PI3K/mTOR pathways in oncology research.
Publications
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